Drugs / Foods that Induce or Inhibit Various Cytochrome P-450 Systems |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Amiodarone | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Amitriptyline | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Anastrozole | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan | 2C8 | Diazepam, Diclofenac, Mephobarbital, Omeprazole, Paclitaxel, Retinoic, Tolbutamide | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Barbiturates | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| 2C19 | Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin |
| 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Broccoli | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Brussel Sprouts | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Buproprion | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Cannabinoids | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Carbamazepine | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| 2C19 | Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin |
| 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Celecoxib | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Charcoal-Broiled Meats | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Chloramphenicol | 2C19 | Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin |
| 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Chlorpheniramine | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Chlorpromazine | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Cimetidine | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| 2C18 | Naproxen, Omeprazole, Proquanil, Propranolol, Piroxicam, Retinoic Acid, Warfarin |
| 2C19 | Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin |
| 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Ciprofloxacin | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Clarithromycin | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Clomipramine | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Clotrimazole | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| 3A5-7 | Cortsol, Ethinyl-Estradiol, Lovastatin, Nifedipine, Quinine, Terfenadine, Testosterone, Triazolam, Vinblastin, Vincristin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Cocaine | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Cyclosporine | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Danazol | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Delavirdine | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Desipramine | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Dexamethasone | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Diclofenac | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Diltiazem | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Disulfram | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| 2E1 | Acetaminophen, Chlorzoxazone, Enflurane, Ethanol, Halothane, Isoflurane, Isoniazid, Ondansetron, Phenol, Ritonavir, Sevoflurane, Tamoxifen, Theophylline |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Doxorubicin | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Efavirenz | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Enoxacin | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Erythromycin | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Ethanol | 2E1 | Acetaminophen, Chlorzoxazone, Enflurane, Ethanol, Halothane, Isoflurane, Isoniazid, Ondansetron, Phenol, Ritonavir, Sevoflurane, Tamoxifen, Theophylline |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Ethosuximide | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Felbamate | 2C19 | Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Flouroquinolones | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Fluconazole | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| 2C19 | Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin |
| 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Fluoxetine | 2C19 | Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin |
| 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Fluphenazine | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Flurbiprofen | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Fluvastatin | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Fluvoxamine | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| 2C19 | Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin |
| 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Glucocorticoids |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Glutethimide |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Grapefruit (juice) | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Griseofulvin |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Haloperidol | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Indinavir |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Indomethicin | 2C19 | Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Insulin | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Isoniazid | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton | 2E1 | Acetaminophen, Chlorzoxazone, Enflurane, Ethanol, Halothane, Isoflurane, Isoniazid, Ondansetron, Phenol, Ritonavir, Sevoflurane, Tamoxifen, Theophylline |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Itraconazole | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Ketoconazone | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| 2C19 | Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin |
| |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| 3A5-7 | Cortsol, Ethinyl-Estradiol, Lovastatin, Nifedipine, Quinine, Terfenadine, Testosterone, Triazolam, Vinblastin, Vincristin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Ketoprofen | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Lansoprazole | 2C19 | Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Levofloxacin | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Lomefloxacin | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Lomustine | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Lovastatin | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Metoclopramide | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Methodone | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Metronidazole | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| 3A5-7 | Cortsol, Ethinyl-Estradiol, Lovastatin, Nifedipine, Quinine, Terfenadine, Testosterone, Triazolam, Vinblastin, Vincristin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Mexiletine | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Mibefradil | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Miconazole |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| 3A5-7 | Cortsol, Ethinyl-Estradiol, Lovastatin, Nifedipine, Quinine, Terfenadine, Testosterone, Triazolam, Vinblastin, Vincristin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Modafinal | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| 2C19 | Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin |
| |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Nafcillin | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Nefazodone | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Nelfinavir |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Nevirapine |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Nicotine | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Norethindrone | 2C19 | Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Norfloxacin | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Norfluoxetine |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Ofloxacin | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Omeprazole | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan | 2C8 | Diazepam, Diclofenac, Mephobarbital, Omeprazole, Paclitaxel, Retinoic, Tolbutamide |
| 2C19 | Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin |
| |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Orphenadrine | 2C19 | Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Paroxetine | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| 2C19 | Bupropion, Cyclophosphamide, Efavirenz, Methadone, Temoxifen |
| 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine | ||
| |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Perphenazine | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Phenobarbital | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan | 2B6 | Bupropion, Cyclophosphamide, Efavirenz, Ifosfamide, Methadone, Tamoxifen | 2C8 | Diazepam, Diclofenac, Mephobarbital, Omeprazole, Paclitaxel, Retinoic, Tolbutamide | |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| 3A5-7 | Cortsol, Ethinyl-Estradiol, Lovastatin, Nifedipine, Quinine, Terfenadine, Testosterone, Triazolam, Vinblastin, Vincristin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Phenylbutazone |
3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Phenytoin | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan | 2B6 | Bupropion, Cyclophosphamide, Efavirenz, Ifosfamide, Methadone, Tamoxifen | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| 3A5-7 | Cortsol, Ethinyl-Estradiol, Lovastatin, Nifedipine, Quinine, Terfenadine, Testosterone, Triazolam, Vinblastin, Vincristin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Prednisone | 2C19 | Bupropion, Cyclophosphamide, Efavirenz, Methadone, Temoxifen |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Primidone | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan | 2B6 | Bupropion, Cyclophosphamide, Efavirenz, Ifosfamide, Methadone, Tamoxifen | 2C8 | Diazepam, Diclofenac, Mephobarbital, Omeprazole, Paclitaxel, Retinoic, Tolbutamide | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| 3A5-7 | Cortsol, Ethinyl-Estradiol, Lovastatin, Nifedipine, Quinine, Terfenadine, Testosterone, Triazolam, Vinblastin, Vincristin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Probenicid | 2C19 | Bupropion, Cyclophosphamide, Efavirenz, Methadone, Temoxifen |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Propafenone | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Propoxyphene | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin | |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Quinidine | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Ranitidine | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Rifampin | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan | 2B6 | Bupropion, Cyclophosphamide, Efavirenz, Ifosfamide, Methadone, Tamoxifen | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton | 2C19 | Bupropion, Cyclophosphamide, Efavirenz, Methadone, Temoxifen | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin | 3A5-7 | Cortsol, Ethinyl-Estradiol, Lovastatin, Nifedipine, Quinine, Terfenadine, Testosterone, Triazolam, Vinblastin, Vincristin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Ritonavir | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan | 2A6 | Nicotine, Ritonavir, Tamoxifen | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton | 2C19 | Bupropion, Cyclophosphamide, Efavirenz, Methadone, Temoxifen | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine | 2E1 | Acetaminophen, Chlorzoxazone, Enflurane, Ethanol, Halothane, Isoflurane, Isoniazid, Ondansetron, Phenol, Ritonavir, Sevoflurane, Tamoxifen, Theophylline | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Saquinavir | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Secobarbital | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Sertindole | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Sertraline | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton | 2C19 | Bupropion, Cyclophosphamide, Efavirenz, Methadone, Temoxifen | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Smoking | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| St. John's Wort | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Sulfamethoxazole-trimethoprim | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Sulfinpyrazone | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Sulfonamides | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Tacrine | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Terbinafine | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Thiotepa | 2B6 | Bupropion, Cyclophosphamide, Efavirenz, Ifosfamide, Methadone, Tamoxifen |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Thioridazine | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Ticlopidine | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan | 2B6 | Bupropion, Cyclophosphamide, Efavirenz, Ifosfamide, Methadone, Tamoxifen | 2C19 | Bupropion, Cyclophosphamide, Efavirenz, Methadone, Temoxifen |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Tobacco | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Tolbutamide | 2C19 | Bupropion, Cyclophosphamide, Efavirenz, Methadone, Temoxifen |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Topiramate | 2C19 | Bupropion, Cyclophosphamide, Efavirenz, Methadone, Temoxifen |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Troglitazone | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton | 2C19 | Bupropion, Cyclophosphamide, Efavirenz, Methadone, Temoxifen | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Troleandomycin | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin | 3A5-7 | Cortsol, Ethinyl-Estradiol, Lovastatin, Nifedipine, Quinine, Terfenadine, Testosterone, Triazolam, Vinblastin, Vincristin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Venlafaxine | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Verapamil | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Vinblastine | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Vinorelbine | 2D6 | Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Zafirlukast | 2C9 | Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Zaleuton | 1A2 | Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan |
| DRUG | INDUCES | INHIBITS | DRUGS EFFECTED |
| Zileuton | 3A4 | Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin |