CYTOCHROME P-450 AND DRUG INTERACTIONS

Drugs / Foods that Induce or Inhibit Various Cytochrome P-450 Systems
and the Drugs that are effected by this Induction or Inhibition.


DRUG INDUCES INHIBITS DRUGS EFFECTED

 
Amiodarone   1A2 Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan
    2C9 Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton
    2D6 Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine
    3A4 Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

 
Amitriptyline   2D6 Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine
   
DRUG INDUCES INHIBITS DRUGS EFFECTED

 
Anastrozole   1A2 Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan
    2C8 Diazepam, Diclofenac, Mephobarbital, Omeprazole, Paclitaxel, Retinoic, Tolbutamide
    2C9 Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

 
Barbiturates 1A2   Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan
  2C19   Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin
  2C9   Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton
  3A4   Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

 
Broccoli 1A2   Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

 
Brussel Sprouts 1A2   Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan

DRUG INDUCES INHIBITS DRUGS EFFECTED

Buproprion   2D6 Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Cannabinoids   3A4 Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Carbamazepine 2C9   Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton
  2C19   Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin
  3A4   Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Celecoxib   2D6 Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

 
Charcoal-Broiled Meats 1A2   Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Chloramphenicol   2C19 Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin
    3A4 Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Chlorpheniramine   2D6 Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine

DRUG INDUCES INHIBITS DRUGS EFFECTED

Chlorpromazine   2D6 Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine
   
DRUG INDUCES INHIBITS DRUGS EFFECTED

Cimetidine   1A2 Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan
    2C9 Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton
    2C18 Naproxen, Omeprazole, Proquanil, Propranolol, Piroxicam, Retinoic Acid, Warfarin
    2C19 Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin
    2D6 Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine
    3A4 Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Ciprofloxacin   1A2 Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan
    3A4 Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Clarithromycin   1A2 Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan
    3A4 Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Clomipramine   2D6 Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine
    3A4 Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
   
DRUG INDUCES INHIBITS DRUGS EFFECTED

Clotrimazole   3A4 Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
    3A5-7 Cortsol, Ethinyl-Estradiol, Lovastatin, Nifedipine, Quinine, Terfenadine, Testosterone, Triazolam, Vinblastin, Vincristin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Cocaine   2D6 Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Cyclosporine   3A4 Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
   
DRUG INDUCES INHIBITS DRUGS EFFECTED

Danazol   3A4 Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
   
DRUG INDUCES INHIBITS DRUGS EFFECTED

Delavirdine   3A4 Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Desipramine   2D6 Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Dexamethasone 2D6   Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine
  3A4   Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Diclofenac   2C9 Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Diltiazem   1A2 Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan
    3A4 Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Disulfram   2C9 Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton
    2E1 Acetaminophen, Chlorzoxazone, Enflurane, Ethanol, Halothane, Isoflurane, Isoniazid, Ondansetron, Phenol, Ritonavir, Sevoflurane, Tamoxifen, Theophylline
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Doxorubicin   2D6 Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Efavirenz 3A4   Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Enoxacin   1A2 Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Erythromycin   1A2 Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan
    3A4 Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Ethanol 2E1   Acetaminophen, Chlorzoxazone, Enflurane, Ethanol, Halothane, Isoflurane, Isoniazid, Ondansetron, Phenol, Ritonavir, Sevoflurane, Tamoxifen, Theophylline
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Ethosuximide 3A4   Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Felbamate   2C19 Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Flouroquinolones   1A2 Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Fluconazole   2C9 Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton
    2C19 Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin

  3A4 Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Fluoxetine   2C19 Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin
    2D6 Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine

  3A4 Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Fluphenazine   2D6 Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Flurbiprofen   2C9 Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Fluvastatin   2C9 Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Fluvoxamine   1A2 Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan
    2C9 Amitriptyline, Carvedilol, Celecoxib, Dapsone, Diclofenac, Dronabinol, Fluoxetine, Fluvoxamine, Glimepiride, Gliizide, Glyburide, Hexobarbital, Ibuprofen, Imipramine, Indomethacin, Irbessartan, Losartan, Mefenamic Acid, Meloxicam, Mirtazapine, Naproxen, Nateglinide, Phenacetin, Piroxicam, Ritonavir, Rosiglitazone, Sildenafil, Sulfamethoxazole, Tamoxifen, Tolbutamide, Torsemide, Warfarin, Zafirlukast, Zileuton
    2C19 Amitriptyline, Carisoprodol, Citalopram, Clomipramine, Cyclophosphamide, Diazepam, Divalproex sodium, Hexobarbital, Imipramine, Indomethacin, Lansoprazole, Mephenytoin, Mephobarbital, Nevirapine, Nilutamide, Omeprazole, Pantoprazole, Phenytoin, Primidone, Progesterone, Proguanil, Propranolol, Ritonavir, Teniposide, Valproic Acid, Warfarin
    2D6 Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine

  3A4 Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Glucocorticoids
3A4   Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Glutethimide
3A4   Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Grapefruit (juice)   1A2 Acetaminophen, Amitriptyline, Caffeine, Clomipramine, Clozapine, Cyclobenzamine, Despiramine, Diazepam, Ethinyl Estradiol, Fluvoxamine, Haloperidol, Imipramine, Isotretinoin (retinoids), Maxiletine, Methadone, Mirtazapine, Naproxen, Nortriptyline, Olanzapine, Ondansetron, Phenacetin, Propafenone, Propranolol, R-Warfarin, Riluzole, Ritonavir, Ropivacaine, Tacrine, Tamoxifen, Theophylline, Verapamil, Warfarin, Zileuton, Zolmitriptan

  3A4 Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Griseofulvin
3A4   Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, Sildenafil, Sirolimus, Simvastatin, Sufentanil, Tacrolimus, Tamoxifen, Taxol, Temazepam, Teniposide, Terfenadine, Testosterone, Theophylline, Tiagabine, Trazodone, Triazolam, Troleandomycin, Verapamil, Vinblastin, Vinca alkaloids, Vincristin, Zaleplon, Zileutin
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Haloperidol   2D6 Amitriptyline, Amphetamine, Atomoxetine, Bisoprolol, Carvedilol, Chlorpheniramine, Chlorpromazine, Clomipramine, Clozapine, Codeine, Cyclobenzaprine, Delaviridine, Desipramine, Dexfenfluramine, Dextromethorphan, Dolasetron, Donepezil, Encainide, Fenfluamine, Flecainide, Fluxetine, Fluphenazine, Fluvoxamine, Haloperidol, Hydrocodone, Hydrocortisone, Imipramine, Indinavir, Labetalol, Lidocaine, Loratadine, Maprotiline, Maxiletine, Meperidine, Methadone, Methamphetamine, Metoclopramide, Metoprolol, Mexiletine, Mirtazapine, Morphine, Nortriptyline, Ondansetron, Oxycodone, Paroxetine, Perpenazine, Phenacetin, Phenformin, Propafenone, Propranolol, Risperidone, Ritonavir, Ropivacaine, Selegiline, Sertindole, Sertraline, Tamoxifen, Thioridazine, Timolol, Tramadol, Trazodone, Tropisetron, Venlafaxine, Yohimbine
 
DRUG INDUCES INHIBITS DRUGS EFFECTED

Indinavir
  3A4 Acetaminophen, Alfentanil, Alprazolam, Amiodarone, Amitriptyline, Amiodipine, Anastrozole, Astemizole, Atovastatin, Bepridil, Buspirone, Busulfan, Cafergot, Caffeine, Cannabinoids, Carbamazepine, Cerivastatin, Chlorpheniramine, Chlorpromazine, Cimetidine, Cisapride, Clarithromycin, Clindamycin, Clomipramine, Clonazepam, Cocaine, Codeine, Cortsol, Cyclonenzaprine, Cyclophosphamide, Cyclosporin, Dapsone, Delavirdine, Dexamethazone, Dextromethorphan, Diazepam, Diltiazem, Disopyramide, Dolasetron, Donepezil, Doxorubicin, Enalapril, Ergot Alkaloids, Erythromycin, Estrogens(oral), Ethinyl-Estradiol, Ethosuximide, Etoposide, Felodipine, Fentanyl, Fexofenadine, Finasteride, Fluconazole, Flutamide, Gleevac, Glyburide, Granisetron, Haloperidol, Hydrocodone, Hydrocortisone, Ifosfamide, Imipramine, Indinavir, Irinotecan, Isotretinoin(retinoids), Isradipine, Itraconazole, Ketoconazole, Lansoprazole, Lidocaine, Loratadine, Losartan, Lovastatin, Methadone, Miconazole, Midazolam, Mirtazapine, Nateglinide, Navalbine, Nefazodone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldpine, Nitrendipine, Ondansetron, Oral-contraceptives, Paclitaxel, Pimozide, Pravastatin, Prednisone, Progesterone, Propafenone, Quinidine, Quinine, R-Warfarin, Rapamycin, Rifabutin, Rifampin, Ritonavir, Salmeterol, Saquinavir, Sertraline, S